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Management of coronary artery disease via simvastatin-loaded novasomes.

Management of coronary artery disease via simvastatin-loaded novasomes.

期刊: Journal of microencapsulation 日期: 2026-03-01 PMID: 42341093 DOI: 10.1080/02652048.2026.2688996 浏览: 28
作者: Fouad AG, Belal A, Yousef Gushgari O, Ahmed Bawaked R, Abdullah Al Shwail F, Abo El-Ela FI
AG, F., A, B., O, Y.G., R, A.B., F, A.A.S., & FI, A.E.E. (2026). Management of coronary artery disease via simvastatin-loaded novasomes.. Journal of microencapsulation. https://doi.org/10.1080/02652048.2026.2688996
AG F, A B, O YG, R AB, F AAS, FI AEE. Management of coronary artery disease via simvastatin-loaded novasomes.. Journal of microencapsulation. 2026; doi: 10.1080/02652048.2026.2688996
AG F, A B, O YG, et al. Management of coronary artery disease via simvastatin-loaded novasomes.[J]. Journal of microencapsulation. 2026. DOI: 10.1080/02652048.2026.2688996.
@article{ag2026,
  author = {Fouad AG and Belal A and Yousef Gushgari O and Ahmed Bawaked R and Abdullah Al Shwail F and Abo El-Ela FI},
  title = {Management of coronary artery disease via simvastatin-loaded novasomes.},
  journal = {Journal of microencapsulation},
  year = {2026},
  doi = {10.1080/02652048.2026.2688996},
  note = {PMID: 42341093},
}
TY  - JOUR
AU  - Fouad AG
AU  - Belal A
AU  - Yousef Gushgari O
AU  - Ahmed Bawaked R
AU  - Abdullah Al Shwail F
AU  - Abo El-Ela FI
TI  - Management of coronary artery disease via simvastatin-loaded novasomes.
T2  - Journal of microencapsulation
PY  - 2026
DO  - 10.1080/02652048.2026.2688996
AN  - PMID:42341093
ER  - 

摘要

BACKGROUND: Simvastatin (SMT) offers protection against diabetes mellitus related to coronary artery disease (DM-CAD) because of its cardioprotective, antioxidant, and anti-inflammatory effects. However, its low bioavailability and poor solubility limit its effectiveness. OBJECTIVE: This research aimed to develop and evaluate a nasal simvastatin-loaded novasomes (S-NOV) to enhance the drug's bioavailability, solubility, and effectiveness in treating DM-CAD. METHODS: The efficacy and bioavailability of the nasal S-NOV formulation were tested in a DM-CAD-induced rat model. RESULTS: The optimal S-NOV formulation demonstrated an 8.31-fold increase in bioavailability, a 4.64-fold enhancement in permeability, and a 4.71-fold increase in drug release. The nasal S-NOV formulation showed superior cardioprotective and antioxidant effects compared to oral SMT in various biomarkers, including lactate dehydrogenase, glutathione, and catalase. Histopathological and toxicology studies confirmed that the nasal S-NOV formulation was effective and safe. CONCLUSION: These findings suggest that nasal S-NOV formulation could be a viable and safe therapy for DM-CAD.

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